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Oxytocin Acetate
EfficacyHigh
Studies45
Participants25,000
StatusAvailable

Oxytocin Acetate

Cys-Tyr-Ile-Gln-Asn-Cys-Pro-Leu-Gly-NH₂

Oxytocin Acetate is a synthetic form of the naturally occurring neuropeptide hormone oxytocin. FDA-approved for obstetric uses including labor induction, augmentation, and postpartum hemorrhage prevention. In research settings, it shows promise for treating autism spectrum disorders and enhancing social cognition through its effects on oxytocin receptors in the brain and peripheral tissues.

Complete Dosing Guide

Quick Reference

0.5-20
Typical Dose
Variable
Frequency
1-6
Half-Life
SubQ
Route

Administration Method

Intravenous infusion, intramuscular injection, or intranasal spray

Step-by-Step Dosing Protocol

Initial
0.5-20 mU/min IV (labor) or 10 IU IM (PPH prevention)
Getting started
Follow gradual escalation approach
Maintenance
Optimized dose
Sustained benefits
Continue at effective dose
Cycling
Break period
Recovery
Take breaks to maintain effectiveness

Dosing Guidelines

Research Protocol

Labor induction begins with 0.5-1 mU/min IV, increasing by 1-2 mU/min every 30-60 minutes until adequate contractions achieved (maximum 20 mU/min). Postpartum hemorrhage prevention uses 10 IU intramuscular immediately after delivery. Treatment of active bleeding employs 10-40 IU in 500-1000mL IV fluid. Research protocols for autism use 24-48 IU intranasal spray daily.

Simple Explanation

For labor, doctors start with a very small amount through an IV and slowly increase it every 30-60 minutes until contractions are strong enough. For preventing bleeding after delivery, one injection is given in the muscle. The amounts are carefully calculated - too little won't work, too much can cause problems, so medical supervision is always required.

Mixing & Injection

Technical Instructions

Primary route is intravenous continuous infusion using controlled infusion pumps for precise dosing during labor. Intramuscular injection in deltoid or gluteal muscle for single-dose applications like PPH prevention. Intranasal spray formulations used in research settings for CNS effects. Subcutaneous administration rarely used clinically but employed in some research protocols.

Step-by-Step Guide

Primary route is intravenous continuous infusion using controlled infusion pumps for precise dosing during labor. Intramuscular injection in deltoid or gluteal muscle for single-dose applications like PPH prevention. Intranasal spray formulations used in research settings for CNS effects. Subcutaneous administration rarely used clinically but employed in some research protocols.

Clinical Administration Guidelines

Injection Protocol

  • Subcutaneous injection per protocol
  • Rotate injection sites
  • Consistent daily timing
  • Follow protocol guidelines

Monitoring Schedule

  • Regular progress monitoring
  • Health parameter monitoring
  • Laboratory monitoring
  • Safety monitoring

Dosage Calculator

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Medical Disclaimer

Oxytocin Acetate is FDA-approved for obstetric uses and requires medical supervision. This information is for educational purposes and should not replace consultation with healthcare providers. Individual results may vary. Proper monitoring is essential during all clinical applications.